List of steroidal antiandrogens

Progesterone derivatives

Abiraterone (CB-7598) = 17-(3-pyridinyl)androsta-5,16-dien-3β-ol
Abiraterone acetate = 17-(3-pyridinyl)androsta-5,16-dien-3β-ol acetate
Benorterone (SKF-7690, FC-612) = 17α-methyl-B-nortestosterone
BOMT (Ro 7-2340) = 6α-bromo-4-oxa-17α-methyl-4,5α-dihydrotestosterone
Delanterone (GBR-21162) = 17β-dehydroxy-1α-methyl-δ¹⁶-testosterone
Dienogest = 17α-cyanomethyl-19-nor-δ⁹⁽¹⁰⁾-testosterone
Epitestosterone = 17α-epitestosterone
Galeterone (TOK-001, VN/124-1) = 17-(1H-benzimidazol-1-yl)androsta-5,16-dien-3β-ol
Metogest (SC-14207) = 16,16-dimethyl-19-nortestosterone
Mifepristone = 11β-[p-(dimethylamino)phenyl]-17-(1-propynyl)-δ⁹-19-nortestosterone
Oxendolone (TSAA-291) = 16β-ethyl-19-nortestosterone
Rosterolone (SH-434, 17α-propylmesterolone) = 1α-methyl-17α-propyl-4,5α-dihydrotestosterone
Topterone (WIN-17665) = 17α-propyltestosterone
Trimethyltrienolone (R-2956, RU-2956) = 2α,2β,17α-trimethyl-19-nor-δ^9,11-testosterone
Zanoterone (WIN-49596) = (5α,17α)-1'-(methylsulfonyl)-1'-H-pregn-20-yno[3,2-c]pyrazol-17-ol

SC-5233 (spirolactone) = 17α-(2-carboxyethyl)testosterone γ-lactone
SC-8109 = 19-norspirolactone
Canrenone (aldadiene) = Δ⁶-spirolactone
Dicirenone (SC-26304) = 7α-carboxyisopropylspirolactone
Drospirenone = 6β,7β:15β,16β-dimethylenespirolactone
Mespirenone (ZK-94679) = Δ¹-7α-acetylthio-15β,16β-methylenespirolactone
Mexrenone (ZK-32055, SC-25152) = 7α-(methoxycarbonyl)spirolactone
Prorenone (SC-23133) = 6α,7α-methylenespirolactone
Spironolactone = 7α-acetylthiospirolactone
Spirorenone (ZK-35973) = Δ¹-6β,7β:15β,16β-dimethylenespirolactone
Spiroxasone = 7α-acetylthiospirolactone with the ketone group removed from the C17α spirolactone ring

9,11-Dehydrocortexolone 17α-butyrate (CB-03-04) = 17α-(butyryloxy)-9,11-didehydrodeoxycorticosterone
Clascoterone (CB-03-01; cortexolone 17α-propionate, 11-deoxycortisol 17α-propionate) = 17α-(propionyloxy)deoxycorticosterone